← Mechanisms of action
Integrin alpha-L/beta-2 (LFA-1)
PROTEIN COMPLEXHomo sapiens
Linked proteins
Drugs acting on this target (3)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| lifitegrast (xiidra) | Antagonist | approved | Small molecule | Integrin alpha-L/beta-2 (LFA-1) antagonist |
| rovelizumab (LeukArrest) | Antagonist | experimental | mAb | Integrin alpha-L/beta-2 (LFA-1) antagonist |
| efalizumab (Raptiva) | Inhibitor | withdrawn | mAb | Integrin alpha-L/beta-2 (LFA-1) inhibitor |