← Mechanisms of action

TACR3

SINGLE PROTEINHomo sapiens
Preferred name: Neurokinin 3 receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (9)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
azd-2624AntagonistexperimentalSmall moleculeTACR3 antagonist
elinzanetantAntagonistapprovedSmall moleculeTACR3 antagonist
fezolinetant (Veozah)AntagonistapprovedSmall moleculeTACR3 antagonist
gsk1144814AntagonistexperimentalSmall moleculeTACR3 antagonist
nt-814AntagonistexperimentalSmall moleculeTACR3 antagonist
osanetantAntagonistexperimentalSmall moleculeTACR3 antagonist
talnetantAntagonistexperimentalSmall moleculeTACR3 antagonist
abcl635InhibitorexperimentalmAbTACR3 inhibitor
sjx-653InhibitorexperimentalSmall moleculeTACR3 inhibitor