← Mechanisms of action
Retinoic acid receptor
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (14)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| adapalene (differin) | Agonist | approved | Small molecule | Retinoic acid receptor agonist |
| cis-retinoic acid | Agonist | experimental | Small molecule | Retinoic acid receptor agonist |
| isotretinoin (Accutane) | Agonist | approved | Small molecule | Retinoic acid receptor agonist |
| n-(4-hydroxyphenyl)all-trans retinamide | Agonist | experimental | Small molecule | Retinoic acid receptor agonist |
| peretinoin | Agonist | experimental | Small molecule | Retinoic acid receptor agonist |
| retinaldehyde | Agonist | experimental | Small molecule | Retinoic acid receptor agonist |
| tac-101 | Agonist | experimental | Small molecule | Retinoic acid receptor agonist |
| tamibarotene | Agonist | experimental | Small molecule | Retinoic acid receptor agonist |
| tazarotene (tazorac) | Agonist | approved | Small molecule | Retinoic acid receptor agonist |
| tretinoin (Retin-A) | Agonist | approved | Small molecule | Retinoic acid receptor agonist |
| trifarotene (Aklief) | Agonist | approved | Small molecule | Retinoic acid receptor agonist |
| vitamin a | Agonist | approved | Small molecule | Retinoic acid receptor agonist |
| zuretinol | Agonist | experimental | Small molecule | Retinoic acid receptor agonist |
| irx-4310 | Antagonist | experimental | Small molecule | Retinoic acid receptor antagonist |