← Mechanisms of action
Hypoxia inducible factors; HIF-1-alpha, HIF-2-alpha
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (3)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| Belzutifan (Welireg) | Antagonist | approved | Small molecule | Hypoxia inducible factors; HIF-1-alpha, HIF-2-alpha antagonist |
| dff332 | Inhibitor | experimental | Small molecule | Hypoxia inducible factors; HIF-1-alpha, HIF-2-alpha inhibitor |
| molidustat | Inhibitor | experimental | Small molecule | Hypoxia inducible factors; HIF-1-alpha, HIF-2-alpha inhibitor |