← Mechanisms of action
EPAS1
SINGLE PROTEINHomo sapiens
Preferred name: Endothelial PAS domain-containing protein 1 ChEMBL ↗
Linked proteins
Drugs acting on this target (7)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ab521 | Inhibitor | experimental | Small molecule | EPAS1 inhibitor |
| Belzutifan (Welireg) | Inhibitor | approved | Small molecule | Endothelial PAS domain-containing protein 1 inhibitor |
| bpi-452080 | Inhibitor | experimental | Small molecule | EPAS1 inhibitor |
| hrs-10516 | Inhibitor | experimental | Small molecule | EPAS1 inhibitor |
| mbm-01 | Inhibitor | experimental | Small molecule | EPAS1 inhibitor |
| nkt2152 | Inhibitor | experimental | Small molecule | EPAS1 inhibitor |
| aro-hif2 | Rnai inhibitor | experimental | Nucleic acid | EPAS1 rnai inhibitor |