← Mechanisms of action
Serine/threonine-protein kinase AKT
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (13)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| afuresertib | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| azd-5672 | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| capivasertib (Truqap) | Inhibitor | approved | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| gsk-690693 | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| ipatasertib | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| ly2780301 | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| miransertib | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| mk-2201 | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| msk-2206 | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| tas0612 | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| triciribine | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| uprosertib | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |
| xl418 | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase AKT inhibitor |