← Mechanisms of action

PLK1

SINGLE PROTEINHomo sapiens
Preferred name: Serine/threonine-protein kinase PLK1 ChEMBL ↗

Linked proteins

Drugs acting on this target (12)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
tkm-080301Antisense inhibitorexperimentalNucleic acidPLK1 antisense inhibitor
bi-2536InhibitorexperimentalSmall moleculePLK1 inhibitor
cafusertibInhibitorexperimentalSmall moleculePLK1 inhibitor
cafusertibInhibitorexperimentalSmall moleculePLK1 inhibitor
cyc140InhibitorexperimentalSmall moleculePLK1 inhibitor
gsk 461364InhibitorexperimentalSmall moleculePLK1 inhibitor
ivx-214InhibitorexperimentalSmall moleculePLK1 inhibitor
mk-1496InhibitorexperimentalSmall moleculePLK1 inhibitor
nms-1286937InhibitorexperimentalSmall moleculePLK1 inhibitor
onvansertibInhibitorexperimentalSmall moleculePLK1 inhibitor
tak-960InhibitorexperimentalSmall moleculePLK1 inhibitor
volasertibInhibitorexperimentalSmall moleculePLK1 inhibitor