← Mechanisms of action

ITGA4

SINGLE PROTEINHomo sapiens
Preferred name: Integrin alpha-4 ChEMBL ↗

Linked proteins

Drugs acting on this target (9)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
axr-159AntagonistexperimentalSmall moleculeITGA4 antagonist
gs-1427AntagonistexperimentalSmall moleculeITGA4 antagonist
ro0506997AntagonistexperimentalSmall moleculeITGA4 antagonist
atl1102Antisense inhibitorexperimentalNucleic acidITGA4 antisense inhibitor
biib107InhibitorexperimentalmAbITGA4 inhibitor
natalizumab (tysabri)InhibitorapprovedmAbITGA4 inhibitor
spy001InhibitorexperimentalmAbITGA4 inhibitor
trk-170InhibitorexperimentalSmall moleculeITGA4 inhibitor
ZaurategrastInhibitorexperimentalSmall moleculeITGA4 inhibitor