← Mechanisms of action
Integrin alpha-4/beta-7
PROTEIN COMPLEXHomo sapiens
Linked proteins
Drugs acting on this target (7)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| firategrast | Antagonist | experimental | Small molecule | Integrin alpha-4/beta-7 antagonist |
| abrilumab | Inhibitor | experimental | mAb | Integrin alpha-4/beta-7 inhibitor |
| ajm347 | Inhibitor | experimental | Small molecule | Integrin alpha-4/beta-7 inhibitor |
| natalizumab (tysabri) | Inhibitor | approved | mAb | Integrin alpha-4/beta-7 inhibitor |
| pn-943 | Inhibitor | experimental | Small molecule | Integrin alpha-4/beta-7 inhibitor |
| ptg-100 | Inhibitor | experimental | Small molecule | Integrin alpha-4/beta-7 inhibitor |
| vedolizumab (entyvio) | Inhibitor | approved | mAb | Integrin alpha-4/beta-7 inhibitor |