← Mechanisms of action
Dual specificity mitogen-activated protein kinase kinase; MEK1/2
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (3)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| rg-7167 | Inhibitor | experimental | Small molecule | Dual specificity mitogen-activated protein kinase kinase; MEK1/2 inhibitor |
| selumetinib (Koselugo) | Inhibitor | approved | Small molecule | Dual specificity mitogen-activated protein kinase kinase; MEK1/2 inhibitor |
| trametinib (mekinist) | Inhibitor | approved | Small molecule | Dual specificity mitogen-activated protein kinase kinase; MEK1/2 inhibitor |