← Mechanisms of action
Sulfonylurea receptor 1, Kir6.2
PROTEIN COMPLEXHomo sapiens
Linked proteins
Drugs acting on this target (11)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| acetohexamide (dymelor) | Blocker | approved | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |
| chlorpropamide (diabinese) | Blocker | approved | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |
| gliclazide | Blocker | experimental | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |
| glimepiride (amaryl) | Blocker | approved | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |
| glipizide (glucotrol) | Blocker | approved | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |
| glyburide (micronase) | Blocker | approved | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |
| mitiglinide (Glufast) | Blocker | experimental | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |
| nateglinide (starlix) | Blocker | approved | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |
| repaglinide (prandin) | Blocker | approved | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |
| tolazamide (tolinase) | Blocker | approved | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |
| tolbutamide (orinase) | Blocker | approved | Small molecule | Sulfonylurea receptor 1, Kir6.2 blocker |