← Mechanisms of action
DRD1
SINGLE PROTEINHomo sapiens
Preferred name: Dopamine D1 receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (24)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ad-2081 | Activator | experimental | Small molecule | DRD1 activator |
| ly3154885 | Activator | experimental | Small molecule | DRD1 activator |
| Mevidalen | Activator | experimental | Small molecule | DRD1 activator |
| dar-100a | Agonist | experimental | Small molecule | DRD1 agonist |
| dihydrexidine | Agonist | experimental | Small molecule | DRD1 agonist |
| fenoldopam (corlopam) | Agonist | approved | Small molecule | DRD1 agonist |
| kdt-3594 | Agonist | experimental | Small molecule | DRD1 agonist |
| lu ae04621 | Agonist | experimental | Small molecule | DRD1 agonist |
| lu af28996 | Agonist | experimental | Small molecule | DRD1 agonist |
| lu ag06479 | Agonist | experimental | Small molecule | DRD1 agonist |
| mni-968 | Agonist | experimental | Small molecule | DRD1 agonist |
| ecopipam | Antagonist | experimental | Small molecule | DRD1 antagonist |
| methylergometrine | Antagonist | approved | Small molecule | DRD1 antagonist |
| nnc-112 | Antagonist | experimental | Small molecule | DRD1 antagonist |
| zotepine | Antagonist | experimental | Small molecule | DRD1 antagonist |
| zuclopenthixol | Antagonist | experimental | Small molecule | DRD1 antagonist |
| zicronapine | Inhibitor | experimental | Small molecule | DRD1 inhibitor |
| asp4345 | Modulator | experimental | Small molecule | DRD1 modulator |
| ucb0022 | Modulator | experimental | Small molecule | DRD1 modulator |
| cvl-871 | Partial agonist | experimental | Small molecule | DRD1 partial agonist |
| pf-06412562 | Partial agonist | experimental | Small molecule | DRD1 partial agonist |
| pf-06669571 | Partial agonist | experimental | Small molecule | DRD1 partial agonist |
| Tavapadon | Partial agonist | experimental | Small molecule | Dopamine D1 receptor partial agonist |
| Mevidalen | Positive allosteric modulator | experimental | Small molecule | Dopamine D1 receptor positive allosteric modulator |