← Mechanisms of action
Neuronal acetylcholine receptor; alpha3/beta4
PROTEIN COMPLEXHomo sapiens
Linked proteins
Drugs acting on this target (6)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| tc-6499 | Agonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha3/beta4 agonist |
| asm-024 | Antagonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha3/beta4 antagonist |
| pentolinium (ansolysen) | Antagonist | approved | Small molecule | Neuronal acetylcholine receptor; alpha3/beta4 antagonist |
| trimethaphan (arfonad) | Antagonist | approved | Small molecule | Neuronal acetylcholine receptor; alpha3/beta4 antagonist |
| mecamylamine (inversine) | Negative allosteric modulator | approved | Small molecule | Neuronal acetylcholine receptor; alpha3/beta4 negative allosteric modulator |
| larazotide acetate | Partial agonist | experimental | Peptide | Neuronal acetylcholine receptor; alpha3/beta4 partial agonist |