← Mechanisms of action
TGFB1
SINGLE PROTEINHomo sapiens
Preferred name: Transforming growth factor beta-1 ChEMBL ↗
Linked proteins
Drugs acting on this target (40)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| dkf-306 | Activator | experimental | Small molecule | TGFB1 activator |
| AGEN 1423 | Antagonist | experimental | mAb | TGFB1 antagonist |
| ak130 | Antagonist | experimental | mAb | TGFB1 antagonist |
| avid200 | Antagonist | experimental | Small molecule | TGFB1 antagonist |
| bj-005 | Antagonist | experimental | mAb | TGFB1 antagonist |
| es014 | Antagonist | experimental | mAb | TGFB1 antagonist |
| PM-8001 | Antagonist | experimental | mAb | TGFB1 antagonist |
| qlf32004 | Antagonist | experimental | mAb | TGFB1 antagonist |
| qls31901 | Antagonist | experimental | mAb | TGFB1 antagonist |
| srk-001 | Antagonist | experimental | mAb | TGFB1 |
| TQ-B2858 | Antagonist | experimental | mAb | TGFB1 antagonist |
| tu2218 | Antagonist | experimental | Small molecule | TGFB1 antagonist |
| stp707 | Antisense inhibitor | experimental | Nucleic acid | TGFB1 antisense inhibitor |
| trk-250 | Antisense inhibitor | experimental | Nucleic acid | TGFB1 antisense inhibitor |
| sb-01 | Blocker | experimental | Peptide | TGFB1 blocker |
| abbv-151 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| ace-1334 | Inhibitor | experimental | Recombinant protein | TGFB1 inhibitor |
| ace-2494 | Inhibitor | experimental | Recombinant protein | TGFB1 inhibitor |
| bca101 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| bintrafusp alfa | Inhibitor | experimental | Recombinant protein | TGFB1 inhibitor |
| cn202 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| fs-8002 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| gc1008 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| hbt-708 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| imc-tr1 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| js201 | Inhibitor | experimental | Recombinant protein | TGFB1 inhibitor |
| jyb1907 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| luspatercept (Reblozyl) | Inhibitor | approved | Recombinant protein | TGFB1 inhibitor |
| ly2382770 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| metelimumab | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| msb0011359c | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| nis793 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| p144 | Inhibitor | experimental | Peptide | TGFB1 inhibitor |
| ro7496353 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| sar439459 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| shr-1701 | Inhibitor | experimental | Recombinant protein | TGFB1 inhibitor |
| SRK-181 | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| Y101D | Inhibitor | experimental | mAb | TGFB1 inhibitor |
| 89zr-gc1008 | Radiopharmaceutical | experimental | mAb | TGFB1 radiopharmaceutical |
| tgfβ-b-15 peptide | Supplementation | experimental | Peptide | TGFB1 supplementation |