← Mechanisms of action

CCR5

SINGLE PROTEINHomo sapiens
Preferred name: C-C chemokine receptor type 5 ChEMBL ↗

Linked proteins

Drugs acting on this target (18)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
adaptavirAntagonistexperimentalSmall moleculeCCR5 antagonist
aplavirocAntagonistexperimentalSmall moleculeCCR5 antagonist
azd-5672AntagonistexperimentalSmall moleculeCCR5 antagonist
bms-813160AntagonistexperimentalSmall moleculeCCR5 antagonist
cenicrivirocAntagonistexperimentalSmall moleculeCCR5 antagonist
incb-9471AntagonistexperimentalSmall moleculeCCR5 antagonist
maraviroc (selzentry)AntagonistapprovedSmall moleculeCCR5 antagonist
ob-002AntagonistexperimentalSmall moleculeCCR5 antagonist
pf-00232798AntagonistexperimentalSmall moleculeCCR5 antagonist
pf-04634817AntagonistexperimentalSmall moleculeCCR5 antagonist
pro-140 monoclonal antibodyAntagonistexperimentalmAbCCR5 antagonist
vicrivirocAntagonistexperimentalSmall moleculeCCR5 antagonist
ccr5mab004InhibitorexperimentalmAbCCR5 inhibitor
hgs-1025InhibitorexperimentalmAbCCR5 inhibitor
leronlimabInhibitorexperimentalmAbCCR5 inhibitor
pro-140 monoclonal antibodyInhibitorexperimentalmAbCCR5 inhibitor
rap103InhibitorexperimentalPeptideCCR5 inhibitor
sb-728mr-tModulatorexperimentalGene therapyCCR5 modulator