← Mechanisms of action

CDK6

SINGLE PROTEINHomo sapiens
Preferred name: Cyclin-dependent kinase 6 ChEMBL ↗

Linked proteins

Drugs acting on this target (33)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
btx-9341DegraderexperimentalSmall moleculeCDK6 degrader
7-hydroxystaurosporineInhibitorexperimentalSmall moleculeCDK6 inhibitor
abemaciclib (verzenio)InhibitorapprovedSmall moleculeCDK6 inhibitor
alvocidibInhibitorexperimentalSmall moleculeCDK6 inhibitor
bpi-1178InhibitorexperimentalSmall moleculeCDK6 inhibitor
bpi-16350InhibitorexperimentalSmall moleculeCDK6 inhibitor
cs3002InhibitorexperimentalSmall moleculeCDK6 inhibitor
dalpiciclibInhibitorexperimentalSmall moleculeCDK6 inhibitor
darcilideInhibitorexperimentalSmall moleculeCDK6 inhibitor
elv001InhibitorexperimentalSmall moleculeCDK6 inhibitor
eth-155008InhibitorexperimentalSmall moleculeCDK6 inhibitor
fcn-437cInhibitorexperimentalSmall moleculeCDK6 inhibitor
g1t28-1InhibitorexperimentalSmall moleculeCDK6 inhibitor
g1t38InhibitorexperimentalSmall moleculeCDK6 inhibitor
gdc-4198InhibitorexperimentalSmall moleculeCDK6 inhibitor
glr2007InhibitorexperimentalSmall moleculeCDK6 inhibitor
hs-10342InhibitorexperimentalSmall moleculeCDK6 inhibitor
LerociclibInhibitorexperimentalSmall moleculeCDK6 inhibitor
nuv-422InhibitorexperimentalSmall moleculeCDK6 inhibitor
pf-06842874InhibitorexperimentalSmall moleculeCDK6 inhibitor
pf-06873600InhibitorexperimentalSmall moleculeCDK6 inhibitor
prt3645InhibitorexperimentalSmall moleculeCDK6 inhibitor
qls12004InhibitorexperimentalSmall moleculeCDK6 inhibitor
rgt-419bInhibitorexperimentalSmall moleculeCDK6 inhibitor
ribociclib (kisqali)InhibitorapprovedSmall moleculeCDK6 inhibitor
sph6516InhibitorexperimentalSmall moleculeCDK6 inhibitor
syh2043InhibitorexperimentalSmall moleculeCDK6 inhibitor
tqb3303InhibitorexperimentalSmall moleculeCDK6 inhibitor
trilaciclib (Cosela)InhibitorapprovedSmall moleculeCyclin-dependent kinase 6 inhibitor
ty-302InhibitorexperimentalSmall moleculeCDK6 inhibitor
tyk-00540InhibitorexperimentalSmall moleculeCDK6 inhibitor
uct-03-008InhibitorexperimentalSmall moleculeCDK6 inhibitor
xh-30002InhibitorexperimentalSmall moleculeCDK6 inhibitor