← Mechanisms of action

TSPO

SINGLE PROTEINHomo sapiens
Preferred name: Translocator protein ChEMBL ↗

Linked proteins

Drugs acting on this target (12)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
da-5216ActivatorexperimentalSmall moleculeTSPO activator
emapunilAgonistexperimentalSmall moleculeTSPO agonist
ssr180575AgonistexperimentalSmall moleculeTSPO agonist
ono-2952AntagonistexperimentalSmall moleculeTranslocator protein antagonist
dpa-713Binding agentexperimentalSmall moleculeTSPO binding agent
pbr28Binding agentexperimentalSmall moleculeTSPO binding agent
ono-2952InhibitorexperimentalSmall moleculeTSPO inhibitor
sf12051InhibitorexperimentalSmall moleculeTSPO inhibitor
tro40303InhibitorexperimentalSmall moleculeTSPO inhibitor
alpidemPartial agonistexperimentalSmall moleculeTSPO partial agonist
11c-er176RadiopharmaceuticalexperimentalRecombinant proteinTSPO radiopharmaceutical
v0251SupplementationexperimentalGene therapyTSPO supplementation