← Mechanisms of action

XPO1

SINGLE PROTEINHomo sapiens
Preferred name: Exportin-1 ChEMBL ↗

Linked proteins

Drugs acting on this target (10)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
selinexor (Xpovio)AntagonistapprovedSmall moleculeXPO1 antagonist
wj01024AntagonistexperimentalSmall moleculeXPO1 antagonist
BIIB100InhibitorexperimentalSmall moleculeXPO1 inhibitor
EltanexorInhibitorexperimentalSmall moleculeXPO1 inhibitor
kpt-330InhibitorexperimentalSmall moleculeXPO1 inhibitor
kpt-8602InhibitorexperimentalSmall moleculeXPO1 inhibitor
sl-801InhibitorexperimentalSmall moleculeXPO1 inhibitor
verdinexorInhibitorexperimentalSmall moleculeXPO1 inhibitor
wj01075InhibitorexperimentalSmall moleculeXPO1 inhibitor
wjb001InhibitorexperimentalSmall moleculeXPO1 inhibitor