← Mechanisms of action

FFAR1

SINGLE PROTEINHomo sapiens
Preferred name: Free fatty acid receptor 1 ChEMBL ↗

Linked proteins

Drugs acting on this target (13)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
cpl207280AgonistexperimentalSmall moleculeFFAR1 agonist
hd-6277AgonistexperimentalSmall moleculeGPR40
idg-16177AgonistexperimentalSmall moleculeFFAR1 agonist
jtt-851AgonistexperimentalSmall moleculeFFAR1 agonist
ly2881835AgonistexperimentalSmall moleculeFFAR1 agonist
ly2922083AgonistexperimentalSmall moleculeFFAR1 agonist
ly2922470AgonistexperimentalSmall moleculeFFAR1 agonist
mk-8666AgonistexperimentalSmall moleculeFFAR1 agonist
shr0534AgonistexperimentalSmall moleculeFFAR1 agonist
venus 20Binding agentexperimentalSmall moleculeFFAR1 binding agent
p11187InhibitorexperimentalSmall moleculeFFAR1 inhibitor
pbi-4050InhibitorexperimentalSmall moleculeFFAR1 inhibitor
fasiglifamPositive allosteric modulatorexperimentalSmall moleculeFFAR1 positive allosteric modulator