← Mechanisms of action
CASR
SINGLE PROTEINHomo sapiens
Preferred name: Calcium sensing receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (11)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| etelcalcetide (parsabiv) | Agonist | approved | Peptide | CASR agonist |
| shr6508 | Agonist | experimental | Small molecule | CASR agonist |
| atf936 | Antagonist | experimental | Small molecule | CASR antagonist |
| encaleret | Antagonist | experimental | Small molecule | CASR antagonist |
| ronacaleret | Antagonist | experimental | Small molecule | CASR antagonist |
| axt914 | Inhibitor | experimental | Small molecule | CASR inhibitor |
| etelcalcetide (parsabiv) | Inhibitor | approved | Peptide | CASR inhibitor |
| norcalcin | Modulator | experimental | Small molecule | CASR modulator |
| asp-7991 | Positive allosteric modulator | experimental | Small molecule | CASR positive allosteric modulator |
| cinacalcet (sensipar) | Positive allosteric modulator | approved | Small molecule | CASR positive allosteric modulator |
| evocalcet | Positive allosteric modulator | experimental | Small molecule | Calcium sensing receptor positive allosteric modulator |