← Mechanisms of action
AURKA
SINGLE PROTEINHomo sapiens
Preferred name: Serine/threonine-protein kinase Aurora-A ChEMBL ↗
Linked proteins
Drugs acting on this target (16)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| xnw34017 | Degrader | experimental | Small molecule | AURKA degrader |
| alisertib | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| at9283 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| bi 831266 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| bi 847325 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| cenisertib | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| enmd 2076 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| ep0042 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| kw2449 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| ly3295668 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| mk-5108 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| mln8054 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| pf-03814735 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| rg1530 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| tas-119 | Inhibitor | experimental | Small molecule | AURKA inhibitor |
| vic-1911 | Inhibitor | experimental | Small molecule | AURKA inhibitor |