← Mechanisms of action
THRB
SINGLE PROTEINHomo sapiens
Preferred name: Thyroid hormone receptor beta-1 ChEMBL ↗
Linked proteins
Drugs acting on this target (19)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| hp515 | Activator | experimental | Small molecule | THRB activator |
| vk2809 | Activator | experimental | Small molecule | THRB activator |
| alg-055009 | Agonist | experimental | Small molecule | THRB agonist |
| asc41 | Agonist | experimental | Small molecule | THRB agonist |
| asc43f | Agonist | experimental | Small molecule | THRB agonist |
| cs060304 | Agonist | experimental | Small molecule | THRB agonist |
| cs060380 | Agonist | experimental | Small molecule | THRB agonist |
| cu-40101 | Agonist | experimental | Small molecule | THRB agonist |
| ecc4703 | Agonist | experimental | Small molecule | THRB agonist |
| eprotirome | Agonist | experimental | Small molecule | THRB agonist |
| hec169584 | Agonist | experimental | Small molecule | THRB agonist |
| kpc000154 | Agonist | experimental | Small molecule | THRB agonist |
| kylo-0603 | Agonist | experimental | Small molecule | THRB agonist |
| mb07811 | Agonist | experimental | Small molecule | THRB agonist |
| mgl-3196 | Agonist | experimental | Small molecule | THRB agonist |
| resmetirom (REZDIFFRA) | Agonist | approved | Small molecule | THRB agonist |
| tern-501 | Agonist | experimental | Small molecule | THRB |
| vk-0214 | Agonist | experimental | Small molecule | THRB agonist |
| hsk31679 | Inhibitor | experimental | Small molecule | THRB inhibitor |