← Mechanisms of action

HMGCR

SINGLE PROTEINHomo sapiens
Preferred name: HMG-CoA reductase ChEMBL ↗

Linked proteins

Drugs acting on this target (9)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
atorvastatin (lipitor)InhibitorapprovedSmall moleculeHMGCR inhibitor
cerivastatin (baycol)InhibitorwithdrawnSmall moleculeHMGCR inhibitor
fluvastatin (lescol)InhibitorapprovedSmall moleculeHMGCR inhibitor
lovastatin (mevacor)InhibitorapprovedSmall moleculeHMGCR inhibitor
pitavastatin (livalo)InhibitorapprovedSmall moleculeHMGCR inhibitor
pravastatin (pravachol)InhibitorapprovedSmall moleculeHMGCR inhibitor
rosuvastatin (crestor)InhibitorapprovedSmall moleculeHMGCR inhibitor
simvastatin (zocor)InhibitorapprovedSmall moleculeHMGCR inhibitor
syn-010InhibitorexperimentalSmall moleculeHMGCR inhibitor