← Mechanisms of action
EDNRB
SINGLE PROTEINHomo sapiens
Preferred name: Endothelin receptor ET-B ChEMBL ↗
Linked proteins
Drugs acting on this target (4)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| darusentan | Antagonist | experimental | Small molecule | EDNRB antagonist |
| enrasentan | Antagonist | experimental | Small molecule | EDNRB antagonist |
| tezosentan | Antagonist | experimental | Small molecule | EDNRB antagonist |
| rg-7636 | Binding agent | experimental | mAb | EDNRB binding agent |