← Mechanisms of action
CHEK1
SINGLE PROTEINHomo sapiens
Preferred name: Serine/threonine-protein kinase Chk1 ChEMBL ↗
Linked proteins
Drugs acting on this target (15)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| pep07 | Antagonist | experimental | Nucleic acid | CHK1 |
| 7-hydroxystaurosporine | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| azd-7762 | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| azd7760 | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| bbi-355 | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| gdc-0425 | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| gdc-0575 | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| ly2880070 | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| mk-8776 | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| pf-477736 | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| prexasertib | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| rabusertib | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| smp3124lp | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| sra737 | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |
| xl844 | Inhibitor | experimental | Small molecule | CHEK1 inhibitor |