← Mechanisms of action
HTR2B
SINGLE PROTEINHomo sapiens
Preferred name: Serotonin 2b (5-HT2b) receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (18)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| cyb004 | Activator | experimental | Small molecule | HTR2B activator |
| am1476 | Antagonist | experimental | Small molecule | HTR2B antagonist |
| Brilaroxazine | Antagonist | experimental | Small molecule | HTR2B antagonist |
| ketanserin | Antagonist | experimental | Small molecule | HTR2B antagonist |
| metadelfene | Antagonist | experimental | Small molecule | HTR2B antagonist |
| methysergide (sansert) | Antagonist | approved | Small molecule | HTR2B antagonist |
| mianserin (Tolvon) | Antagonist | experimental | Small molecule | HTR2B antagonist |
| s1ra | Antagonist | experimental | Small molecule | HTR2B antagonist |
| sarpogrelate | Antagonist | experimental | Small molecule | HTR2B antagonist |
| spn-810 | Antagonist | experimental | Small molecule | HTR2B antagonist |
| vabicaserin | Antagonist | experimental | Small molecule | HTR2B antagonist |
| viloxazine (Qelbree) | Antagonist | approved | Small molecule | HTR2B antagonist |
| xc101-d13h | Antagonist | experimental | Small molecule | HTR2B antagonist |
| xc130-a10h | Antagonist | experimental | Small molecule | HTR2B antagonist |
| am1030 | Inhibitor | experimental | Small molecule | HTR2B inhibitor |
| amap102 | Inhibitor | experimental | Small molecule | HTR2B inhibitor |
| kt110 | Inhibitor | experimental | Small molecule | HTR2B inhibitor |
| methylergometrine | Partial agonist | approved | Small molecule | HTR2B partial agonist |