← Mechanisms of action
DRD5
SINGLE PROTEINHomo sapiens
Preferred name: Dopamine D5 receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (7)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ad-2081 | Activator | experimental | Small molecule | DRD5 activator |
| dihydrexidine | Agonist | experimental | Small molecule | DRD5 agonist |
| hec113995pa | Inhibitor | experimental | Small molecule | DRD5 inhibitor |
| cvl-871 | Partial agonist | experimental | Small molecule | DRD5 partial agonist |
| pf-06412562 | Partial agonist | experimental | Small molecule | DRD5 partial agonist |
| pf-06669571 | Partial agonist | experimental | Small molecule | DRD5 partial agonist |
| Tavapadon | Partial agonist | experimental | Small molecule | Dopamine D5 receptor partial agonist |