← Mechanisms of action
PDGFRA
SINGLE PROTEINHomo sapiens
Preferred name: Platelet-derived growth factor receptor alpha ChEMBL ↗
Linked proteins
Drugs acting on this target (20)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| avapritinib (Ayvakit) | Antagonist | approved | Small molecule | PDGFRA antagonist |
| olaratumab (lartruvo) | Antagonist | approved | mAb | PDGFRA antagonist |
| sorafenib (nexavar) | Antagonist | approved | Small molecule | PDGFRA antagonist |
| 3d011-08 | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| 89zr-dfosq-olaratumab | Inhibitor | experimental | mAb | PDGFRA inhibitor |
| aiv007 | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| amuvatinib | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| anrotenib | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| avapritinib (Ayvakit) | Inhibitor | approved | Small molecule | Platelet-derived growth factor receptor alpha inhibitor |
| cbt-004 | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| fn-1501 | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| kanitinib | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| nb003 | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| olaratumab (lartruvo) | Inhibitor | approved | mAb | PDGFRA inhibitor |
| radotinib | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| ripretinib (Qinlock) | Inhibitor | approved | Small molecule | Platelet-derived growth factor receptor alpha inhibitor |
| Seralutinib | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| subutinib | Inhibitor | experimental | Small molecule | PDGFRA inhibitor |
| sunitinib (sutent) | Inhibitor | approved | Small molecule | Platelet-derived growth factor receptor alpha inhibitor |
| tovetumab | Inhibitor | experimental | mAb | PDGFRA inhibitor |