← Mechanisms of action
MC1R
SINGLE PROTEINHomo sapiens
Preferred name: Melanocortin receptor 1 ChEMBL ↗
Linked proteins
Drugs acting on this target (10)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| resomelagon | Activator | experimental | Small molecule | MC1R activator |
| afamelanotide (Scenesse) | Agonist | approved | Peptide | Melanocortin receptor 1 agonist |
| asp3291 | Agonist | experimental | Peptide | MC1R agonist |
| bremelanotide (Vyleesi) | Agonist | approved | Peptide | MC1R agonist |
| Dersimelagon | Agonist | experimental | Small molecule | MC1R agonist |
| kd101 | Agonist | experimental | Small molecule | MC1R agonist |
| modimelanotide | Agonist | experimental | Small molecule | MC1R agonist |
| pl8177 | Agonist | experimental | Peptide | MC1R agonist |
| mtc896 | Inhibitor | experimental | Small molecule | MC1R inhibitor |
| nyh100p | Inhibitor | experimental | Small molecule | MC1R inhibitor |