← Mechanisms of action
S1PR1
SINGLE PROTEINHomo sapiens
Preferred name: Sphingosine 1-phosphate receptor Edg-1 ChEMBL ↗
Linked proteins
Drugs acting on this target (23)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| apd-334 | Agonist | experimental | Small molecule | S1PR1 agonist |
| asp4058 | Agonist | experimental | Small molecule | S1PR1 agonist |
| ethoximod | Agonist | experimental | Small molecule | S1PR1 agonist |
| etrasimod (Velsipity) | Agonist | approved | Small molecule | S1PR1 agonist |
| krp-203 | Agonist | experimental | Small molecule | S1PR1 agonist |
| mocravimod | Agonist | experimental | Small molecule | Sphingosine 1-phosphate receptor Edg-1 agonist |
| pf-04629991 | Agonist | experimental | Small molecule | S1PR1 agonist |
| ponesimod (Ponvory) | Agonist | approved | Small molecule | S1PR1 agonist |
| proximod | Agonist | experimental | Small molecule | S1PR1 agonist |
| sar247799 | Agonist | experimental | Small molecule | S1PR1 agonist |
| scd-044 | Agonist | experimental | Small molecule | S1PR1 agonist |
| siponimod (Mayzent) | Agonist | approved | Small molecule | S1PR1 agonist |
| cenerimod | Inhibitor | experimental | Small molecule | S1PR1 inhibitor |
| gsk2018682 | Inhibitor | experimental | Small molecule | S1PR1 inhibitor |
| bms-986104 | Modulator | experimental | Small molecule | S1PR1 modulator |
| cenerimod | Modulator | experimental | Small molecule | Sphingosine 1-phosphate receptor Edg-1 modulator |
| etrasimod (Velsipity) | Modulator | approved | Small molecule | Sphingosine 1-phosphate receptor Edg-1 modulator |
| lc51-0255 | Modulator | experimental | Small molecule | S1PR1 modulator |
| LC51-0255 | Modulator | experimental | Small molecule | S1PR1 modulator |
| mocravimod | Modulator | experimental | Small molecule | S1PR1 modulator |
| opl-002 | Modulator | experimental | Small molecule | S1PR1 modulator |
| ozanimod (Zeposia) | Modulator | approved | Small molecule | Sphingosine 1-phosphate receptor Edg-1 modulator |
| vtx002 | Modulator | experimental | Small molecule | S1PR1 modulator |