← Mechanisms of action
HTR3A
SINGLE PROTEINHomo sapiens
Preferred name: Serotonin 3a (5-HT3a) receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (20)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| pumosetrag | Agonist | experimental | Small molecule | HTR3A agonist |
| alosetron (lotronex) | Antagonist | approved | Small molecule | HTR3A antagonist |
| cvn058 | Antagonist | experimental | Small molecule | HTR3A antagonist |
| ddp225 | Antagonist | experimental | Small molecule | HTR3A antagonist |
| dolasetron (anzemet) | Antagonist | approved | Small molecule | HTR3A antagonist |
| granisetron (kytril) | Antagonist | approved | Small molecule | HTR3A antagonist |
| hrs-5817 | Antagonist | experimental | Small molecule | HTR3A antagonist |
| metoclopramide (reglan) | Antagonist | approved | Small molecule | HTR3A antagonist |
| ondansetron (zofran) | Antagonist | approved | Small molecule | HTR3A antagonist |
| palonosetron (aloxi) | Antagonist | approved | Small molecule | HTR3A antagonist |
| renzapride | Antagonist | experimental | Small molecule | HTR3A antagonist |
| tak-058 | Antagonist | experimental | Small molecule | HTR3A antagonist |
| vortioxetine (trintellix) | Antagonist | approved | Small molecule | HTR3A antagonist |
| itasetron | Inhibitor | experimental | Small molecule | HTR3A inhibitor |
| lerisetron | Inhibitor | experimental | Small molecule | HTR3A inhibitor |
| litoxetine | Inhibitor | experimental | Small molecule | HTR3A inhibitor |
| lx1031 | Inhibitor | experimental | Small molecule | HTR3A inhibitor |
| ramosetron | Inhibitor | experimental | Small molecule | HTR3A inhibitor |
| tropisetron | Inhibitor | experimental | Small molecule | HTR3A inhibitor |
| smp-100 | Partial agonist | experimental | Small molecule | HTR3A partial agonist |