← Mechanisms of action
PTGER2
SINGLE PROTEINHomo sapiens
Preferred name: Prostanoid EP2 receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (10)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| alprostadil (prostin) | Agonist | approved | Small molecule | PTGER2 agonist |
| cp-533,536 | Agonist | experimental | Small molecule | PTGER2 agonist |
| evatanepag | Agonist | experimental | Small molecule | Prostanoid EP2 receptor agonist |
| omidenepag (Omlonti) | Agonist | approved | Small molecule | PTGER2 agonist |
| sar366234 | Agonist | experimental | Small molecule | PTGER2 agonist |
| simenepag isopropyl | Agonist | experimental | Small molecule | PTGER2 agonist |
| taprenepag | Agonist | experimental | Small molecule | Prostanoid EP2 receptor agonist |
| pf-04418948 | Antagonist | experimental | Small molecule | PTGER2 antagonist |
| mbf-362 | Inhibitor | experimental | Small molecule | PTGER2 inhibitor |
| tpst-1495 | Inhibitor | experimental | Small molecule | PTGER2 inhibitor |