← Mechanisms of action
GHSR
SINGLE PROTEINHomo sapiens
Preferred name: Ghrelin receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (16)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ac01 | Agonist | experimental | Small molecule | GHSR agonist |
| anamorelin | Agonist | experimental | Small molecule | GHSR agonist |
| ghrelin | Agonist | experimental | Peptide | GHSR agonist |
| ghrp-3 | Agonist | experimental | Vaccine | GHSR agonist |
| ibutamoren | Agonist | experimental | Small molecule | GHSR agonist |
| macimorelin (Macrilen) | Agonist | approved | Small molecule | GHSR agonist |
| relamorelin | Agonist | experimental | Peptide | GHSR agonist |
| tabimorelin | Agonist | experimental | Small molecule | GHSR agonist |
| tzp-102 | Agonist | experimental | Small molecule | GHSR agonist |
| ulimorelin | Agonist | experimental | Small molecule | GHSR agonist |
| liver-enriched antimicrobial peptide 2 | Antagonist | experimental | Peptide | GHSR antagonist |
| gs3-007 | Inhibitor | experimental | Small molecule | GHSR inhibitor |
| leap2 hormone | Inhibitor | experimental | Peptide | GHSR inhibitor |
| al-53817 | Inverse agonist | experimental | Small molecule | GHSR inverse agonist |
| pf-5190457 | Inverse agonist | experimental | Small molecule | GHSR inverse agonist |
| cp-424,391 | Supplementation | experimental | Small molecule | GHSR supplementation |