← Mechanisms of action
NFKB1
SINGLE PROTEINHomo sapiens
Preferred name: Nuclear factor NF-kappa-B p105 subunit ChEMBL ↗
Linked proteins
Drugs acting on this target (12)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| tepilamide | Activator | experimental | Small molecule | NFKB1 activator |
| amg0103 | Inhibitor | experimental | Nucleic acid | NFKB1 inhibitor |
| avenanthramides | Inhibitor | experimental | Botanical | NFKB1 inhibitor |
| diepalrestat choline | Inhibitor | experimental | Small molecule | NFKB1 inhibitor |
| dimethyl sulfone | Inhibitor | experimental | Small molecule | NFKB1 inhibitor |
| Eucalyptol (listerine) | Inhibitor | experimental | Small molecule | NFKB1 inhibitor |
| heptex | Inhibitor | experimental | Small molecule | NFKB1 inhibitor |
| iguratimod | Inhibitor | experimental | Small molecule | NFKB1 inhibitor |
| nf-kappab decoy | Inhibitor | experimental | Recombinant protein | NFKB1 inhibitor |
| ortd-1 | Inhibitor | experimental | Small molecule | NFKB1 inhibitor |
| xp23829 | Inhibitor | experimental | Small molecule | NFKB1 inhibitor |
| hypoestoxide | Modulator | experimental | Small molecule | NFKB1 modulator |