← Mechanisms of action

OPRD1

SINGLE PROTEINHomo sapiens
Preferred name: Delta opioid receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (15)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
adl 5747AgonistexperimentalSmall moleculeOPRD1 agonist
adl5859AgonistexperimentalSmall moleculeOPRD1 agonist
axomadolAgonistexperimentalSmall moleculeOPRD1 agonist
azd-2327AgonistexperimentalSmall moleculeOPRD1 agonist
azd7268AgonistexperimentalSmall moleculeOPRD1 agonist
dalarginAgonistexperimentalSmall moleculeOPRD1 agonist
dynorphin 1-13AgonistexperimentalPeptideOPRD1 agonist
heroinAgonistexperimentalSmall moleculeOPRD1 agonist
ketobemidone (Ketogan)AgonistexperimentalSmall moleculeOPRD1 agonist
metenkefalinAgonistexperimentalSmall moleculeOPRD1 agonist
norbuprenorphineAgonistexperimentalSmall moleculeOPRD1 agonist
ThienorphineAgonistexperimentalSmall moleculeOPRD1 agonist
naloxolAntagonistexperimentalSmall moleculeOPRD1 antagonist
cutamesineInhibitorexperimentalSmall moleculeOPRD1 inhibitor
samidorphan (Lybalvi)Partial agonistapprovedSmall moleculeDelta opioid receptor partial agonist