← Mechanisms of action
Kinesin-1 heavy chain/ Tyrosine-protein kinase receptor RET
CHIMERIC PROTEINHomo sapiens
Linked proteins
Drugs acting on this target (2)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| pralsetinib (Gavreto) | Inhibitor | approved | Small molecule | Kinesin-1 heavy chain/ Tyrosine-protein kinase receptor RET inhibitor |
| Selpercatinib (Retevmo) | Inhibitor | approved | Small molecule | Kinesin-1 heavy chain/ Tyrosine-protein kinase receptor RET inhibitor |