← Mechanisms of action

Proto-oncogene tyrosine-protein kinase receptor Ret /Nuclear receptor coactivator 4 fusion protein

CHIMERIC PROTEINHomo sapiens

Linked proteins

Drugs acting on this target (2)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
pralsetinib (Gavreto)AntagonistapprovedSmall moleculeProto-oncogene tyrosine-protein kinase receptor Ret /Nuclear receptor coactivator 4 fusion protein antagonist
Selpercatinib (Retevmo)AntagonistapprovedSmall moleculeProto-oncogene tyrosine-protein kinase receptor Ret /Nuclear receptor coactivator 4 fusion protein antagonist