← Mechanisms of action
CRHR1
SINGLE PROTEINHomo sapiens
Preferred name: Corticotropin releasing factor receptor 1 ChEMBL ↗
Linked proteins
Drugs acting on this target (8)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| emicerfont | Antagonist | experimental | Small molecule | CRHR1 antagonist |
| ono-2333ms | Antagonist | experimental | Small molecule | CRHR1 antagonist |
| pexacerfont | Antagonist | experimental | Small molecule | CRHR1 antagonist |
| ssr-125543 | Antagonist | experimental | Small molecule | CRHR1 antagonist |
| verucerfont | Antagonist | experimental | Small molecule | CRHR1 antagonist |
| Antalarmin | Inhibitor | experimental | Small molecule | CRHR1 inhibitor |
| gsk586529 | Inhibitor | experimental | Small molecule | CRHR1 inhibitor |
| hm17321 | Inhibitor | experimental | Small molecule | CRHR1 inhibitor |