← Mechanisms of action

GRM5

SINGLE PROTEINHomo sapiens
Preferred name: Metabotropic glutamate receptor 5 ChEMBL ↗

Linked proteins

Drugs acting on this target (15)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
d-aspartateActivatorexperimentalSmall moleculeGRM5 activator
dasolampanel etibutilAntagonistexperimentalSmall moleculeGRM5 antagonist
fenobamAntagonistexperimentalSmall moleculeGRM5 antagonist
mavoglurantAntagonistexperimentalSmall moleculeGRM5 antagonist
az12713580InhibitorexperimentalSmall moleculeGRM5 inhibitor
adx10059ModulatorexperimentalSmall moleculeGRM5 modulator
azd-2066ModulatorexperimentalSmall moleculeGRM5 modulator
basimglurantModulatorexperimentalSmall moleculeGRM5 modulator
dipraglurantModulatorexperimentalSmall moleculeGRM5 modulator
get 73ModulatorexperimentalSmall moleculeGRM5 modulator
ro5011232ModulatorexperimentalSmall moleculeGRM5 modulator
ro6806127ModulatorexperimentalSmall moleculeGRM5 modulator
azd-2516Negative allosteric modulatorexperimentalSmall moleculeGRM5 negative allosteric modulator
stx107Negative allosteric modulatorexperimentalSmall moleculeGRM5 negative allosteric modulator
abp688RadiopharmaceuticalexperimentalSmall moleculeGRM5 radiopharmaceutical