← Mechanisms of action
SETD2
SINGLE PROTEINHomo sapiens
Preferred name: Histone-lysine N-methyltransferase SETD2 ChEMBL ↗
Linked proteins
Drugs acting on this target (3)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| hydralazine (apresoline) | Activator | approved | Small molecule | SETD2 activator |
| hec53856 | Inhibitor | experimental | Small molecule | SETD2 inhibitor |
| akb-4924 | Stabiliser | experimental | Small molecule | SETD2 stabiliser |