← Mechanisms of action
Keap1/Nrf2
PROTEIN-PROTEIN INTERACTIONHomo sapiens
Linked proteins
Drugs acting on this target (2)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| diroximel (Vumerity) | Agonist | approved | Small molecule | Keap1/Nrf2 agonist |
| bardoxolone | Inhibitor | experimental | Small molecule | Keap1/Nrf2 inhibitor |