← Mechanisms of action

OXTR

SINGLE PROTEINHomo sapiens
Preferred name: Oxytocin receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (12)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
carbetocin (Pabal)AgonistexperimentalSmall moleculeOXTR agonist
deuterated oxytocinAgonistexperimentalSmall moleculeOXTR agonist
fe-202767AgonistexperimentalSmall moleculeOXTR agonist
merotocinAgonistexperimentalPeptideOXTR agonist
oxytocin (syntocinon)AgonistapprovedPeptideOXTR agonist
Atosiban (tractocile)AntagonistexperimentalSmall moleculeOXTR antagonist
barusibanAntagonistexperimentalSmall moleculeOXTR antagonist
epelsibanAntagonistexperimentalSmall moleculeOXTR antagonist
ix-01AntagonistexperimentalSmall moleculeOXTR antagonist
nolasibanAntagonistexperimentalSmall moleculeOXTR antagonist
relcovaptanAntagonistexperimentalSmall moleculeOXTR antagonist
retosibanAntagonistexperimentalSmall moleculeOXTR antagonist