zalypsis

Animal productexperimental

Clinical trial activity

3 trials · 8 clinical orgs · 0 marketing orgs

Phase 1
1
Phase 2
2
Phase 3
0
Phase 4
0

Earliest trial started May 1, 2006 (NCT00359294)

Timeline

2000s

  1. Jan 1, 2006

    Earliest Phase 1 Sponsor(trial)

  2. Jan 1, 2009

    Earliest Phase 2 Sponsor(trial)

Indications

Mechanism of action

  • DNACROSS-LINKING AGENT

    DNA cross-linking agent

Chemistry & pharmacology

Oral

No

Parenteral

No

Topical

No

Also known as

  • n-((5-(acetyloxy)-6,6a,7,13,14,16-hexahydro-8,14-dihydroxy-9-methoxy-4,10,17-trimethyl-7,13-imino-12h-1,3-dioxolo(7,8)isoquino(3,2-b)(3)benzazocin-16-yl)methyl)-3-(3-(trifluoromethyl)phenyl)-2e-propenamide
  • n-(((6as,7r,13s,14s,16r)-5-(acetyloxy)-6,6a,7,13,14,16-hexahydro-8,14-dihydroxy-9-methoxy-4,10,17-trimethyl-7,13-imino-12h-1,3-dioxolo(7,8)isoquino(3,2-b)(3)benzazocin-16-yl)methyl)-3-(3-(trifluoromethyl)phenyl)-2e-propenamide
  • pm00104
  • pm 00104
  • pm-00104
  • zalypsis
  • zalypsis
  • zalypsis
  • zalypsis

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT01222767Phase 2Dec 1, 2010Centre Leon Berard, Istituto Clinico Humanitas - Rozzano (MI), Italy, PharmaMar, St. Jude Children's Hospital, University of Bologna, University of Milan, University of Washington
NCT00900562Phase 2Aug 1, 2009PharmaMar
NCT00359294Phase 1May 1, 2006PharmaMar, Temple University
Showing 3 of 3 trials
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Organizations

Research & Development (8)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
PharmaMarFor profit3322006
Centre Leon BerardAcademic/Hospital1012010
Istituto Clinico Humanitas - Rozzano (MI), ItalyAcademic/Hospital1012010
St. Jude Children's HospitalAcademic/Hospital1012010
Temple UniversityAcademic/Hospital1012006
University of BolognaAcademic/Hospital1012010
University of MilanAcademic/Hospital1012010
University of WashingtonAcademic/Hospital1012010
8 organizations
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