Aspartyl-alanyl-diketopiperazine

Trade name: Ampion

Small moleculeexperimental

Clinical trial activity

14 trials · 1 clinical orgs · 0 marketing orgs

Phase 1
5
Phase 2
10
Phase 3
7
Phase 4
0

Earliest trial started Mar 1, 2013 (NCT01839331)

Timeline

2010s

  1. Jan 1, 2013

    Earliest Phase 3 Sponsor(trial)

  2. Jan 1, 2014

    Earliest Phase 1 Sponsor(trial)

2020s

  1. Jan 1, 2021

    Earliest Phase 2 Sponsor(trial)

Indications

Mechanism of action

  • Unspecified targetOTHER

    Immunomodulation

  • UnclearUnclear

    Unclear unclear

Chemistry & pharmacology

Loading structure…

SMILES

C[C@@H]1NC(=O)[C@H](CC(=O)O)NC1=O
Mol. weight
186.17 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Single Stereoisomer
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • ampion
  • ampion

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT04880161Phase 1May 31, 2021Ampio Pharmaceuticals. Inc.
NCT04839965Phase 2May 31, 2021Ampio Pharmaceuticals. Inc.
NCT04868890Phase 2Apr 30, 2021Ampio Pharmaceuticals. Inc.
NCT04606784Phase 1Oct 28, 2020Ampio Pharmaceuticals. Inc.
NCT04456452Phase 1Jul 27, 2020Ampio Pharmaceuticals. Inc.
NCT03988023Phase 3Jun 24, 2019Ampio Pharmaceuticals. Inc.
NCT03349645Phase 3Dec 8, 2017Ampio Pharmaceuticals. Inc.
NCT03182686Phase 3Jun 19, 2017Ampio Pharmaceuticals. Inc.
NCT02762760Phase 1May 1, 2016Ampio Pharmaceuticals. Inc.
NCT02556710Phase 3Sep 1, 2015Ampio Pharmaceuticals. Inc.
NCT02242435Phase 3Sep 1, 2014Ampio Pharmaceuticals. Inc.
NCT02184156Phase 1/Phase 2 (Phase 2)Jun 1, 2014Ampio Pharmaceuticals. Inc.
NCT02024529Phase 3Dec 1, 2013Ampio Pharmaceuticals. Inc.
NCT01839331Phase 3Mar 1, 2013Ampio Pharmaceuticals. Inc.
Showing 14 of 14 trials
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Organizations

Research & Development (1)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Ampio Pharmaceuticals. Inc.For profit141432013
1 organizations
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