131 iodine

Small moleculeexperimental

Iodide I-131 (as Sodium iodide I-131) is a radioisotopic drug used for the treatment and palliation of thyroid malignancy. Therapeutic solutions of Sodium Iodide-131 are indicated for the treatment of hyperthyroidism and thyroid carcinomas that take up iodine. Palliative effects may be observed in patients with advanced thyroid malignancy if the metastatic lesions take up iodine. It is also indicated for use in performance of the radioactive iodide (RAI) uptake test to evaluate thyroid function. Taken orally, sodium iodide I-131 is rapidly absorbed and distributed within the extracellular fluid of the body. The iodide is concentrated in the thyroid via the sodium/iodide symporter, and subsequently oxidized to iodine. The destruction of thyroidal tissue is achieved by the beta emission of sodium iodide I-131. — NCATS

Clinical trial activity

15 trials · 24 clinical orgs · 0 marketing orgs

Phase 1
2
Phase 2
10
Phase 3
4
Phase 4
0

Earliest trial started Jan 31, 2000 (NCT00115895)

Timeline

2000s

  1. Jan 1, 2000

    Earliest Phase 3 Sponsor(trial)

  2. Jan 1, 2005

    Earliest Phase 1 Sponsor(trial)

2010s

  1. Jan 1, 2011

    Earliest Phase 2 Sponsor(trial)

Indications

Mechanism of action

  • Unspecified targetRadiodepletion

    radiodepletion

Chemistry & pharmacology

Loading structure…

SMILES

[131I-]
Mol. weight
130.906124168 g/mol

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • 131 iodine
  • sun-131

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT05142904Phase 3Nov 17, 2021Free University of Amsterdam, Rijnstate Hospital, University of Twente, ZonMw: The Netherlands Organisation for Health Research and Development
NCT04871139N/AApr 8, 2021National Cancer Institute (NCI), University of Texas at Houston
NCT04447183Phase 2Dec 1, 2020Suzhou Zelgen Biopharmaceuticals Co.,Ltd
NCT03248440Phase 3Jul 31, 2017Senju Pharmaceuticals
NCT03109847Phase 2Jan 5, 2017Thomas Jefferson University
NCT02493712Phase 2Jan 1, 2016Holy Stone Healthcare Co., Ltd, inVentiv, Istituto Clinico Humanitas - Rozzano (MI), Italy
NCT02338648Phase 2Oct 1, 2014Senju Pharmaceuticals
NCT02114619N/AMay 1, 2013Mashhad University of Medical Sciences
NCT01601093Phase 2Nov 1, 2011Nanjing Medical University, Xiangbei Welman Pharmaceutical Co., Ltd
NCT01360177N/AJul 1, 2010Stanford University
NCT00549523Phase 1/Phase 2 (Phase 2)Apr 1, 2008National Center for Complementary and Integrative Health (NCCIH), Office of Dietary Supplements (ODS), University of Missouri
NCT01150318N/AJan 1, 2006University of Paris
NCT00673010Phase 1Mar 1, 2005Cornell University, Institut Gustave Roussy
NCT00196729Phase 3Dec 1, 2001Genzyme
NCT00115895Phase 3Jan 31, 2000University of Helsinki
Showing 15 of 15 trials
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Organizations

Research & Development (24)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Senju PharmaceuticalsFor profit2222014
Cornell UniversityAcademic/Hospital1112005
Free University of AmsterdamAcademic/Hospital1012021
GenzymeFor profit1112001
Holy Stone Healthcare Co., LtdFor profit1112016
Institut Gustave RoussyAcademic/Hospital1012005
inVentivFor profit1012016
Istituto Clinico Humanitas - Rozzano (MI), ItalyAcademic/Hospital1012016
Mashhad University of Medical SciencesAcademic/Hospital1112013
Nanjing Medical UniversityAcademic/Hospital1012011
National Cancer Institute (NCI)Government1012021
National Center for Complementary and Integrative Health (NCCIH)Government1012008
Office of Dietary Supplements (ODS)Government1012008
Rijnstate HospitalAcademic/Hospital1112021
Stanford UniversityAcademic/Hospital1112010
Suzhou Zelgen Biopharmaceuticals Co.,LtdFor profit1112020
Thomas Jefferson UniversityAcademic/Hospital1112017
University of HelsinkiAcademic/Hospital1112000
University of MissouriAcademic/Hospital1112008
University of ParisAcademic/Hospital1112006
24 organizations
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