tartaric acid

Small moleculeapproved

Approved

Aug 7, 1985

Tartaric acid is a white, crystalline organic acid that occurs naturally in many fruits, most notably in grapes but also in tamarinds, bananas, avocados, and citrus. Its salt, potassium bitartrate, commonly known as cream of tartar, develops naturally in the process of fermentation. Potassium bitartrate is commonly mixed with sodium bicarbonate and is sold as baking powder used as a leavening agent in food preparation. The acid itself is added to foods as an antioxidant E334 and to impart its distinctive sour taste. Naturally occurring tartaric acid is a useful raw material in organic synthesis. Tartaric acid, an alpha-hydroxy-carboxylic acid, is diprotic and aldaric in acid characteristics and is a dihydroxyl derivative of succinic acid. — Wikipedia

Clinical trial activity

8 trials · 12 clinical orgs · 2 marketing orgs

Phase 1
0
Phase 2
3
Phase 3
2
Phase 4
1

Earliest trial started Jan 2, 2007 (NCT00754767)

Timeline

1980s

  1. Aug 7, 1985

    Avon Products — Earliest FDA Approval

  2. Aug 7, 1985

    Mallinckrodt — NDA Secondary Org

  3. Aug 7, 1985

    Avon Products — NDA Secondary Org

  4. Aug 7, 1985

    Avon Products — NDA Organization

2020s

  1. Jan 1, 2021

    Earliest Phase 2 Sponsor(trial)

  2. Jan 1, 2024

    Earliest Phase 3 Sponsor(trial)

Indications

Mechanism of action

  • Unspecified targetOTHER

    Radiographic contrast agent

    Tartaric acid and sodium bicarbonate generate carbon dioxide following oral administration. Carbon dioxide extends the stomach and provides a negative contrast medium during double contrast radiography.

  • Unspecified targetUnclear

    Unclear

Combination products

Approval history

  • approvedAug 7, 1985

Chemistry & pharmacology

Loading structure…

SMILES

O=C(O)[C@@H](O)[C@H](O)C(=O)O
Mol. weight
150.09 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Single Stereoisomer
Inorganic
No
Polymer
No
Availability
Discontinued

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • aluminum tartrate
  • ammonium tartrate
  • anhydrous sodium tartrate
  • calcium tartrate
  • calcium tartrate tetrahydrate
  • dextrotartaric acid
  • disodium l-tartrate
  • disodium tartrate
  • e334
  • e334
  • l-tartrate
  • l-tartrate
  • mn(iii) tartrate
  • potassium tartrate
  • potassium tartrate
  • potassium tartrate
  • (r*,r*)-(+-)-2,3-dihydroxybutanedioic acid, monoammonium monosodium salt
  • (r,r)-tartaric acid
  • seignette salt
  • sodium ammonium tartrate
  • sodium potassium tartrate
  • sodium potassium tartrate
  • sodium potassium tartrate
  • sodium tartrate
  • sodium tartrate
  • sodium tartrate
  • sodium tartrate
  • sodium tartrate dihydrate
  • stannous tartrate
  • tartaric acid
  • tartaric acid
  • tartaric acid
  • tartaric acid
  • tartaric acid
  • tartaric acid
  • tartaric acid
  • tartaric acid, ammonium sodium salt, (1:1:1) salt, (r*,r*)-(+-)-isomer
  • tartaric acid, calcium salt, (r-r*,r*)-isomer
  • tartaric acid, monoammonium salt, (r-(r*,r*))-isomer
  • tartaric acid, ((r*,r*)-(+-))-isomer
  • tartaric acid, (r-(r*,r*))-isomer
  • tartaric acid, (r*,s*)-isomer
  • tartaric acid, (s-(r*,r*))-isomer
  • tartrate
  • threaric acid

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT06285799Phase 3Mar 5, 2024Nemysis Ltd, RDC Clinical Pty Ltd
NCT05950841Phase 3Jan 1, 2024RDC Clinical Pty Ltd
NCT06524596N/AJan 1, 2022Wuhan Children's Hospital
NCT05446961Phase 2Mar 1, 2021Hospital Espanhol, SENAI CIMATEC
NCT05022732N/AMay 5, 2020Fondazione Casemiro Mondino, University of Pavia
NCT04375696Phase 4Apr 24, 2020Certmedica International GmbH, University of Pavia
NCT03212677N/AMay 17, 2017Bill and Melinda Gates Foundation, Tufts University
NCT00754767N/AJan 2, 2007HealthPartners Institute, Park Nicollet
Showing 8 of 8 trials
Page 1 / 1

Organizations

Research & Development (12)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
RDC Clinical Pty LtdFor profit2112024
University of PaviaAcademic/Hospital2122020
Bill and Melinda Gates FoundationAcademic/Hospital1012017
Certmedica International GmbHFor profit1112020
Fondazione Casemiro MondinoAcademic/Hospital1012020
HealthPartners InstituteAcademic/Hospital1112007
Hospital EspanholAcademic/Hospital1012021
Nemysis LtdFor profit1112024
Park NicolletAcademic/Hospital1012007
SENAI CIMATECAcademic/Hospital1112021
Tufts UniversityAcademic/Hospital1112017
Wuhan Children's HospitalAcademic/Hospital1112022
12 organizations
Page 1 / 1

Marketing (3)

OrganizationOrg typeRelationshipDate
Avon ProductsFor profitNDA2Aug 7, 1985
Avon ProductsFor profitNDAAug 7, 1985
MallinckrodtFor profitNDA2Aug 7, 1985