diquafosol

Small moleculeexperimental

Diquafosol is a pharmaceutical drug for the treatment of dry eye disease. It was approved for use in Japan in 2010. It is formulated as a 3% ophthalmic solution of the tetrasodium salt. — Wikipedia

Clinical trial activity

14 trials · 12 clinical orgs · 0 marketing orgs

Phase 1
2
Phase 2
5
Phase 3
3
Phase 4
2

Earliest trial started Aug 15, 2017 (NCT03640351)

Timeline

2010s

  1. Jan 1, 2017

    Earliest Phase 1 Sponsor(trial)

2020s

  1. Jan 1, 2020

    Earliest Phase 3 Sponsor(trial)

  2. Jan 1, 2022

    Earliest Phase 2 Sponsor(trial)

Indications

Approved for

Mechanism of action

Chemistry & pharmacology

Oral

No

Parenteral

No

Topical

No

Sources

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT06903884Phase 3Dec 30, 2025The University of Hong Kong
NCT07097922N/AAug 1, 2025He Eye Hospital
NCT06852105N/AFeb 28, 2025He Eye Hospital
NCT06427031Phase 3Jul 14, 2023Taejoon Pharm Co., Ltd.
NCT07297316Phase 4Oct 3, 2022Korea University, Kukje Pharma
NCT06146881Phase 2Oct 2, 2022Santen Inc., University of Indonesia
NCT05383612N/AAug 5, 2022
NCT06560580N/ANov 15, 2021Tianjin Eye Hospital
NCT05346783Phase 1/Phase 2 (Phase 2)Oct 14, 2021Taejoon Pharm Co., Ltd., Yonsei University
NCT04668118Phase 4Jan 1, 2021Peking University
NCT04548427Phase 3Aug 18, 2020Chong Kun Dang Pharmaceutical, Pusan National University
NCT05456061N/AAug 1, 2018Yonsei University
NCT03216096Phase 1Sep 8, 2017Santen Inc.
NCT03640351N/AAug 15, 2017Yonsei University
Showing 14 of 14 trials
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Organizations

Research & Development (12)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Yonsei UniversityAcademic/Hospital3222017
He Eye HospitalAcademic/Hospital2212025
Santen Inc.For profit2122017
Taejoon Pharm Co., Ltd.For profit2222021
Chong Kun Dang PharmaceuticalFor profit1112020
Korea UniversityAcademic/Hospital1112022
Kukje PharmaFor profit1012022
Peking UniversityAcademic/Hospital1112021
Pusan National UniversityAcademic/Hospital1012020
The University of Hong KongAcademic/Hospital1112025
Tianjin Eye HospitalAcademic/Hospital1112021
University of IndonesiaAcademic/Hospital1112022
12 organizations
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