Lisaftoclax
Small moleculeexperimental
Clinical trial activity
23 trials · 19 clinical orgs · 0 marketing orgs
Phase 1
16
Phase 2
13
Phase 3
4
Phase 4
0
Earliest trial started Aug 7, 2018 (NCT03537482)
Timeline
Indications
Studied for
- Amyloidosis · Phase 1/Phase 2
- Breast Neoplasms · Phase 1/Phase 2
- Hematologic Neoplasms · Early Phase 1
- Leukemia · Phase 1
- Leukemia, Lymphocytic, Chronic, B-Cell · Phase 3
- Leukemia, Myelogenous, Chronic, BCR-ABL Positive · Phase 1
- Leukemia, Myeloid, Acute · Phase 3
- Leukemia, Prolymphocytic, T-Cell · Phase 1
- Lupus Erythematosus, Systemic · Phase 1/Phase 2
- Lymphoma, Non-Hodgkin · Phase 1
- Multiple Myeloma · Phase 1/Phase 2
- Myelodysplastic Syndromes · Phase 3
- Neoplasms · Phase 1/Phase 2
- Neuroblastoma · Phase 1
- Pharmacokinetics · Phase 1
- Precursor Cell Lymphoblastic Leukemia-Lymphoma · Phase 1
- Waldenstrom Macroglobulinemia · Phase 1
Mechanism of action
- Apoptosis regulator Bcl-2INHIBITOR
BCL2 inhibitor
Chemistry & pharmacology
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- ChEMBLCHEMBL4650374 ↗
Clinical trials
| NCT ID | Phase | Start date | Sponsor(s) |
|---|---|---|---|
| NCT07255963 | Phase 2 | Nov 30, 2025 | Soochow University |
| NCT07272499 | Phase 2 | Sep 10, 2025 | Anhui Medical University, Central South University, Fudan University, Fujian Medical University, Jiao Tong University, Shandong University, Tongji University, Wenzhou Medical University |
| NCT06641414 | Phase 3 | Oct 31, 2024 | Ascentage Pharma Group Inc., Peking University, University of Texas at Houston |
| NCT06401603 | Phase 1 | Aug 6, 2024 | Ascentage Pharma Group Inc., University of Texas at Houston |
| NCT06389292 | Phase 3 | Jun 11, 2024 | Ascentage Pharma Group Inc., Chinese Academy of Medical Sciences, Zhejiang University |
| NCT06319456 | Phase 3 | Apr 7, 2024 | Ascentage Pharma Group Inc., Chinese Academy of Medical Sciences |
| NCT06182969 | Phase 1/Phase 2 (Phase 2) | Dec 31, 2023 | Ascentage Pharma Group Inc., Government of China, Jiao Tong University |
| NCT06104566 | Phase 3 | Dec 20, 2023 | Ascentage Pharma Group Inc. |
| NCT05701306 | Phase 1 | Mar 23, 2023 | Ascentage Pharma Group Inc., Government of China, Sun Yat-Sen University |
| NCT05517616 | Phase 1 | Sep 18, 2022 | Ascentage Pharma Group Inc., Soochow University |
| NCT05495035 | Phase 1 | Sep 1, 2022 | China Academy of Chinese Medical Sciences, Chinese Academy of Medical Sciences |
| NCT05147467 | Phase 2 | Jan 31, 2022 | Ascentage Pharma Group Inc., Nanjing Medical University |
| NCT04946864 | Phase 1/Phase 2 (Phase 2) | Aug 13, 2021 | Ascentage Pharma Group Inc. |
| NCT04964518 | Phase 1 | Jul 30, 2021 | Ascentage Pharma Group Inc. |
| NCT04942067 | Phase 1/Phase 2 (Phase 2) | Jun 1, 2021 | Ascentage Pharma Group Inc. |
| NCT04674514 | Phase 1/Phase 2 (Phase 2) | Apr 13, 2021 | Ascentage Pharma Group Inc., Government of China |
| NCT04496349 | Phase 1 | Dec 1, 2020 | Ascentage Pharma Group Inc. |
| NCT04501120 | Phase 1/Phase 2 (Phase 2) | Sep 28, 2020 | Ascentage Pharma Group Inc., Government of China, Suzhou Yasheng Pharmaceutical Co., Ltd |
| NCT04494503 | Phase 1/Phase 2 (Phase 2) | Aug 31, 2020 | Ascentage Pharma Group Inc. |
| NCT04260217 | Phase 1 | Jan 30, 2020 | Ascentage Pharma Group Inc. |
Showing 20 of 23 trials
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Organizations
Research & Development (19)
| Organization | Org type | Trials | As lead sponsor | Phases | Earliest year |
|---|---|---|---|---|---|
| Ascentage Pharma Group Inc. | For profit | 20 | 19 | 3 | 2018 |
| Chinese Academy of Medical Sciences | Academic/Hospital | 4 | 0 | 2 | 2019 |
| Government of China | Government | 4 | 0 | 2 | 2020 |
| Jiao Tong University | Academic/Hospital | 2 | 1 | 1 | 2023 |
| Soochow University | Academic/Hospital | 2 | 1 | 2 | 2022 |
| University of Texas at Houston | Academic/Hospital | 2 | 1 | 2 | 2024 |
| Anhui Medical University | Academic/Hospital | 1 | 0 | 1 | 2025 |
| Central South University | Academic/Hospital | 1 | 0 | 1 | 2025 |
| China Academy of Chinese Medical Sciences | Academic/Hospital | 1 | 1 | 1 | 2022 |
| Fudan University | Academic/Hospital | 1 | 0 | 1 | 2025 |
| Fujian Medical University | Academic/Hospital | 1 | 0 | 1 | 2025 |
| Nanjing Medical University | Academic/Hospital | 1 | 0 | 1 | 2022 |
| Peking University | Academic/Hospital | 1 | 0 | 1 | 2024 |
| Shandong University | Academic/Hospital | 1 | 0 | 1 | 2025 |
| Sun Yat-Sen University | Academic/Hospital | 1 | 0 | 1 | 2023 |
| Suzhou Yasheng Pharmaceutical Co., Ltd | For profit | 1 | 0 | 1 | 2020 |
| Tongji University | Academic/Hospital | 1 | 0 | 1 | 2025 |
| Wenzhou Medical University | Academic/Hospital | 1 | 0 | 1 | 2025 |
| Zhejiang University | Academic/Hospital | 1 | 0 | 1 | 2024 |
19 organizations
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