chlorphenoxamine
Small moleculeexperimental
Chlorphenoxamine is an antihistamine and anticholinergic used as an antipruritic and was formerly used in the sympathomimetic treatment of parkinsonism. Histamine receptor H1 antagonist. Chlorphenoxamine is used to treat Allergic conditions, it is reported as an ingredient of Systral in Germany, Malta, Portugal, Thailand, Turkey. — NCATS
Clinical trial activity
0 trials · 0 clinical orgs · 0 marketing orgs
Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0
Indications
Approved for
Mechanism of action
- Histamine H1 receptorANTAGONIST
HRH1 antagonist
Chlorphenoxamine is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
Chemistry & pharmacology
Loading structure…
SMILES
CN(C)CCOC(C)(c1ccccc1)c1ccc(Cl)cc1- Mol. weight
- 303.83 g/mol
- Lipinski Ro5
- Pass
- Rule of 3
- No
- Chirality
- Racemic Mixture
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- ChEMBLCHEMBL2110774 ↗
- WikipediaChlorphenoxamine ↗
- NCATS3UVD77BP8R ↗
- ChEMBLCHEMBL2105980 ↗
Also known as
- chlorphenoxamine
- chlorphenoxamine
- chlorphenoxamine
- chlorphenoxamine
- chlorphenoxamine
- chlorphenoxamine
- chlorphenoxamine
- chlorphenoxamine hcl
- chlorphenoxamine hcl
- chlorphenoxamine hydrochloride
- chlorphenoxamine hydrochloride
- chlorphenoxamine hydrochloride
- chlorphenoxamine hydrochloride
- chlorphenoxamine hydrochloride
- chlorphenoxamine hydrochloride
- phenoxene
- phenoxene
- systral
- systral
- systral