pyroglutamic acid

Small moleculeexperimental

Clinical trial activity

7 trials · 8 clinical orgs · 0 marketing orgs

Phase 1
4
Phase 2
2
Phase 3
0
Phase 4
1

Earliest trial started Jan 1, 2001 (NCT00040456)

Timeline

2000s

  1. Jan 1, 2001

    Earliest Phase 2 Sponsor(trial)

  2. Jan 1, 2004

    Earliest Phase 1 Sponsor(trial)

Indications

Approved for

Mechanism of action

  • Unspecified targetSupplementation

    supplementation

Chemistry & pharmacology

Loading structure…

SMILES

O=C1CC[C@@H](C(=O)O)N1
Mol. weight
129.12 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Single Stereoisomer
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • (−)-2-pyrrolidone-5-carboxylic acid
  • (−)-2-pyrrolidone-5-carboxylic acid
  • glutimic acid
  • glutimic acid
  • l-5-pyrrolidone-2-carboxylic acid
  • l-5-pyrrolidone-2-carboxylic acid
  • l-pyroglutamic acid
  • l-pyroglutamic acid
  • l-pyrrolidone carboxylic acid
  • l-pyrrolidone carboxylic acid
  • magnesium pidolate
  • magnesium pidolate
  • magnesium pidolate
  • magnesium pidolate
  • magnesium pidolate
  • magnesium pidolate
  • pca
  • pca
  • pidolic acid
  • pidolic acid
  • pidolic acid
  • pidolic acid magnesium salt
  • pyroglutamic acid
  • pyroglutamic acid
  • pyroglutamic acid
  • (s)-(−)-2-pyrrolidone-5-carboxylic acid
  • (s)-(−)-2-pyrrolidone-5-carboxylic acid
  • (s)-pyroglutamic acid
  • (s)-pyroglutamic acid

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT05374343Phase 1May 5, 2022Sichuan University, Sunshine Lake Pharma Co., Ltd.
NCT05427682Phase 1Apr 19, 2022Sunshine Lake Pharma Co., Ltd.
NCT05109078Phase 1Dec 31, 2021Soochow University, Sunshine Lake Pharma Co., Ltd.
NCT01181830Phase 4Feb 1, 2010University of Verona
NCT00532883Phase 2Jan 1, 2007National Heart, Lung, and Blood Institute (NHLBI), St. Jude Children's Hospital
NCT00143572Phase 1Nov 1, 2004St. Jude Children's Hospital
NCT00040456Phase 2Jan 1, 2001Baylor University, Harvard University
Showing 7 of 7 trials
Page 1 / 1

Organizations

Research & Development (8)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Sunshine Lake Pharma Co., Ltd.For profit3312021
St. Jude Children's HospitalAcademic/Hospital2222004
Baylor UniversityAcademic/Hospital1112001
Harvard UniversityAcademic/Hospital1012001
National Heart, Lung, and Blood Institute (NHLBI)Government1012007
Sichuan UniversityAcademic/Hospital1012022
Soochow UniversityAcademic/Hospital1012021
University of VeronaAcademic/Hospital1112010
8 organizations
Page 1 / 1